Product Name: PT-141 (Bremelanotide)
Product Ingredients: Bremelanotide
PT-141 is considered as a synthetic aphrodisiac. Alternatively to Viagra and Cialis, it has no influence upon the vascular system, but directly increases sexual desire. PT-141 activates the melanocortin receptors MC1R and MC4R in the central nervous system, modulates inflammation and reduces the restriction in blood supply to the tissues. PT-141 is a deaminated derivative and metabolite of Melanotan II. PT-141 also acts as an agonist. PT-141 has proved its safeness and efficiency on a broad range of patients.
PT-141 is indicated to treat sexual problems both in men (erectile dysfunction or impotence) and women (sexual arousal disorder). The drug is also prescribed for the medication of hemorrhagic shock and reperfusion injury.
Contraindications and Cautions:
It is contradicted to use more than 1 dose per day, specifically 4mg by nasal spray and 2mg by injection. There are no other strict contradictions for the medication. However it is recommended to consult with the doctor before using the product.
PT-141 (Bremelanotide) is considered to be much safer compared to Viagra or Cialis. However, as all other medicine it might be the reason of several adverse reactions to occur, such as nausea, decreased appetite; flushing of the face and increased blood pressure. The last one should not cause discomfort for healthy individuals. Injectable PT-141 is considered not to have this particular minor effect.
The recommended dose of PT-141 is the same for male and female patients.
The injectable PT-141 should be administrated in the quantity of 2mg per injection and 5 x 2mg injections per vial. The amount to inject will be the following:
1ml of water for dissolving provides then 2mg = 0.2ml (or 20 units on the Insulin Syringe);
2ml of water for mixing provides 2mg = 0.4ml (or 40 units);
3ml of water for mixing provides 2mg = 0.6ml (or 60 units).
PT-141 Nasal Spray recommended dose is 4mg and 5 x 4mg per nasal kit. The inserted amount is the following: the mix of 1ml of water per vial will provide with 4mg = 8 sprays assuming the nasal spray kit as 20mg (2 vials) of PT-141.
Bacteriostatic water, sterile water or sterile saline (0.09nacl) might be used for dilution.
The injectable PT-141 is administrated by subcutaneous injection into fat (thigh, buttock or stomach) with an insulin syringe.
The effects of PT-141 Nasal Spray occur within 1-2 hours for libido enhancement and inducing erections in males. Injectable PT-141 will take at least 2-3 hours before the product to begin taking effect. PT-141 has a long term effect up to 72 hours.
In case of a failed dose it is recommended to administrate it as soon as possible. If it is a time for the next dose, the patient should skip the missed one and return to his regular dosage plan. It is contradicted to double the dose to catch up.
If an overdose occurs the patient should immediately contact his physician or seek an emergent medical help.
There is no notice of the product's interference with other medicine. However, it is recommended to consult with the physician before the PT-141's medication.
The product should be kept at the refrigerator. The dissolved vials might be stored at the refrigerator for a period of 1 month.